SCHEMBL5802115

SCHEMBL5802115

Cc1ccc2c(c1)C(CC1=CNC(=S)[N]1)CC2

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
HTR2B P41595 1/20 0.32
KDM2B Q8NHM5 1/20 0.31
IDO1 P14902 1/20 0.30
TRPV1 Q8NER1 1/20 0.30
MTNR1A P48039 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5800695 0.85 ESR1 (0.37) ESR1ESR2DRD2DRD1HTR2C
SCHEMBL5799245 0.85 ESR1 (0.37) ESR1ESR2HTR2CSLC6A4KDM2B
SCHEMBL5802150 0.82 HTR6 (0.47) ESR1ESR2IDO1MTNR1A
SCHEMBL5798616 0.78 ESR1 (0.37) ESR1ESR2SLC6A4KDM2BIDO1
SCHEMBL1340040 0.71 ESR1 (0.38) ESR1ESR2DRD2DRD1HTR2C
SCHEMBL5801954 0.70 MTNR1A (0.50) MTNR1A
SCHEMBL6185230 0.68
SCHEMBL28748207 0.68 ESR1 (0.36) ESR1ESR2DRD2DRD1HTR2C
SCHEMBL5799895 0.66 HTR6 (0.47) ESR1ESR2IDO1MTNR1A
SCHEMBL28746633 0.66 ESR1 (0.36) ESR1ESR2DRD2DRD1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006036404-A1 4-(SUBSTITUTED CYCLOALKYLMETHYL) IMIDAZOLE-2-THONES, 4-(SUBSTITUTED CYCLOALKENYLMETHYL) IMIDAZOLE-2-THIONES, 4-(SUBSTITUTED CYLOALKYLMETHYL) IMIDAZOL-2-ONES, 4-(SUBSTITUTED CYCLOALKENYLMETHYL) IMIDAZOL-2-ONES AND RELATED COMPOUNDS ALLERGAN, INC. (US) 2006-04-06 WO disclosed