SCHEMBL5799773

SCHEMBL5799773

COC(=O)c1ccc(C=C(CNc2ccc3ccc(OC)cc3c2)COc2cccc3ccccc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 2/20 0.43
ALDH1A1 P00352 4/20 0.42
HPGD P15428 3/20 0.42
POLB P06746 2/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 4/20 0.42
RAPGEF3 O95398 2/20 0.41
KDM4E B2RXH2 3/20 0.40
GCGR P47871 1/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
BLM P54132 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DAPK1 P53355 1/20 0.39
PIM3 Q86V86 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
PLAU P00749 1/20 0.39
GLA P06280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5799769 1.00 P2RX3 (0.43) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5797822 0.93 MEN1 (0.46) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5796297 0.92 P2RX3 (0.52) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5809911 0.89 HPGD (0.44) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5809908 0.89 HPGD (0.44) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5796119 0.88 MAPT (0.47) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5810269 0.86 ALDH1A1 (0.43) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5810275 0.86 ALDH1A1 (0.43) P2RX3ALDH1A1HPGDPOLBKMT2A
SCHEMBL5819819 0.84 P2RX3 (0.43) P2RX3ALDH1A1KMT2AMEN1MAPT
SCHEMBL5814020 0.83 ALPL (0.45) P2RX3ALDH1A1HPGDKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006025683-A1 ARYLAMINOMETHYL PROPENYL BENZHYDROXYAMID DERIVATIVES WITH INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-03-09 WO disclosed