SCHEMBL5799798

SCHEMBL5799798

NC(=O)Oc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.70
NR4A1 P22736 1/20 0.64
NR4A2 P43354 1/20 0.64
NR4A3 Q92570 1/20 0.64
LMNA P02545 1/20 0.61
CYP1A2 P05177 1/20 0.61
PTGS1 P23219 1/20 0.61
SLC6A2 P23975 1/20 0.61
CYP2C19 P33261 1/20 0.61
PTGS2 P35354 1/20 0.61
SLC6A3 Q01959 1/20 0.61
HIF1A Q16665 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
MAOB P27338 3/20 0.60
GAA P10253 1/20 0.59
MAPT P10636 1/20 0.59
MAOA P21397 1/20 0.59
RAB9A P51151 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5249598 0.85 KMT2A (0.65) PARP10NR4A2MAOBMAOASMN1; SMN2
SCHEMBL6634107 0.84 PARP10 (0.68) PARP10NR4A1NR4A2NR4A3LMNA
SCHEMBL5843729 0.83 LTA4H (0.63) PARP10NR4A1NR4A2NR4A3LMNA
SCHEMBL1068959 0.82 MAOB (0.70) PARP10NR4A1NR4A2NR4A3LMNA
SCHEMBL4432728 0.82 PARP10 (0.70) PARP10NR4A1NR4A2NR4A3LMNA
SCHEMBL13719578 0.82 NR4A1 (0.64) PARP10NR4A1NR4A2NR4A3LMNA
SCHEMBL119689 0.82 PARP10 (1.00) PARP10NR4A1NR4A2NR4A3LMNA
Diphenan SCHEMBL667724 0.81 PLA2G10 (0.58) PARP10LMNAL3MBTL1SRD5A2LTA4H
SCHEMBL28694024 0.81 PARP10 (0.64) PARP10NR4A1NR4A2NR4A3LMNA
SCHEMBL1395785 0.81 PARP10 (0.68) PARP10NR4A1NR4A2NR4A3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113336704-B Danshensu derivative and preparation method and medical application thereof 上海大学 2022-10-11 CN disclosed
CN-113336704-A Danshensu derivative and preparation method and medical application thereof 上海大学 2021-09-03 CN disclosed
WO-2006060082-A1 TRICYCLIC COMPOUNDS, PREPARATION THEREOF AND USE THEREOF AS CHOLINESTERASE ACTIVITY INHIBITORS THE GOVERNMENT OF THE U.S.A. as represented by THE SEC., DEPT. OF HEALTH & HUMAN SERVICES, NATIONAL INSTITUTES OF HEALTH (US) 2006-06-08 WO disclosed