SCHEMBL580033

SCHEMBL580033

CC(c1ccccc1)[C@](C(=O)O)(c1ccccc1)N1CCC(C)(O)CC1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 13/20 0.39
OPRK1 P41145 13/20 0.39
OPRL1 P41146 13/20 0.39
OPRD1 P41143 12/20 0.39
CYP2D6 P10635 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK1 P28482 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL305262 1.00 OPRM1 (0.39) OPRM1OPRK1OPRL1OPRD1CYP2D6
SCHEMBL305263 1.00 OPRM1 (0.39) OPRM1OPRK1OPRL1OPRD1CYP2D6
SCHEMBL304094 0.88 OPRL1 (0.53) OPRM1OPRK1OPRL1OPRD1
SCHEMBL304095 0.88 OPRL1 (0.53) OPRM1OPRK1OPRL1OPRD1
SCHEMBL571259 0.68 OPRM1 (0.38) OPRM1OPRK1OPRL1OPRD1CYP2D6
SCHEMBL1316739 0.68 GAA (0.38) OPRK1CYP1A2CYP2C9CYP2C19MAPK1
SCHEMBL1316741 0.68 GAA (0.38) OPRK1CYP1A2CYP2C9CYP2C19MAPK1
SCHEMBL571260 0.68 OPRM1 (0.38) OPRM1OPRK1OPRL1OPRD1CYP2D6
SCHEMBL303920 0.67 LMNA (0.63) OPRM1OPRK1OPRL1OPRD1CYP2D6
SCHEMBL2707046 0.67 LMNA (0.63) OPRM1OPRK1OPRL1OPRD1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417126-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2012-02-15 EP disclosed
WO-2011075439-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-06-23 WO disclosed
WO-2011059887-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed
WO-2011059850-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed