SCHEMBL5800822

SCHEMBL5800822

Cc1c([C@H](C)C(=O)OC(C)C)c2c(F)c(O)c(F)cc2n1C(=O)c1ccc(F)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.35
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NR1H4 Q96RI1 5/20 0.33
ESR1 P03372 1/20 0.32
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
AR P10275 1/20 0.32
PTPN11 Q06124 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
CHRNA1 P02708 1/20 0.31
CHRNG P07510 1/20 0.31
CHRNB1 P11230 1/20 0.31
CHRNB2 P17787 1/20 0.31
SLC6A2 P23975 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5800820 1.00 PTGS2 (0.35) PTGS2MEN1KMT2ANR1H4ESR1
SCHEMBL5813347 0.92 PTGS2 (0.34) PTGS2PTPN11AKR1C3AKR1C2
SCHEMBL5813350 0.92 PTGS2 (0.34) PTGS2PTPN11AKR1C3AKR1C2
SCHEMBL5800314 0.91 PTGS2 (0.32) PTGS2MEN1KMT2AAKR1C3AKR1C2
SCHEMBL5797831 0.90 PTGS2 (0.34) PTGS2PTPN11AKR1C3AKR1C2
SCHEMBL5797833 0.90 PTGS2 (0.34) PTGS2PTPN11AKR1C3AKR1C2
SCHEMBL5813216 0.90 ALDH1A1 (0.35) PTGS2MEN1KMT2ANR1H4AKR1C3
SCHEMBL5813215 0.90 ALDH1A1 (0.35) PTGS2MEN1KMT2ANR1H4AKR1C3
SCHEMBL5813477 0.89 ELANE (0.35) PTGS2MEN1KMT2ANR1H4CHRNA1
SCHEMBL5813474 0.89 ELANE (0.35) PTGS2MEN1KMT2ANR1H4CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed