SCHEMBL5800900

SCHEMBL5800900

CCOCC(=O)Nc1c(Cl)nc2ccccc2c1NCCNC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 4/20 0.47
KDM4E B2RXH2 6/20 0.46
POLB P06746 2/20 0.46
GLA P06280 1/20 0.46
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 2/20 0.44
HTT P42858 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPK1 P28482 1/20 0.44
TSHR P16473 1/20 0.43
GAA P10253 2/20 0.42
LMNA P02545 1/20 0.40
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40
MEN1 O00255 1/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14950200 0.90 TOP2A (0.48) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL1456618 0.88 BCHE (0.46) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL1457271 0.84 KDM4E (0.45) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL1457334 0.84 TOP2A (0.45) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL24879683 0.83 KDM4E (0.44) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL7637380 0.83 KDM4E (0.44) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL8571971 0.82 KDM4E (0.43) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL20766797 0.77 GAA (0.47) TOP2AKDM4EPOLBGLAALDH1A1
SCHEMBL31709349 0.76 ALDH1A1 (0.38) ALDH1A1RAB9ABCHEACHEKMT2A
SCHEMBL1457309 0.76 ACP1 (0.37) TOP2AKDM4EPOLBALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006065280-A2 ISOXAZOLE, DIHYDROISOXAZOLE, AND OXADIAZOLE SUBSTITUTED IMIDAZO RING COMPOUNDS AND METHODS 3M INNOVATIVE PROPERTIES COMPANY (US) 2006-06-22 WO disclosed