SCHEMBL5801978

SCHEMBL5801978

CCCc1ccc(C2[N]CCC2c2cn(Cc3ccc(C(F)(F)F)cc3)c3ccccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC5A1 P13866 6/20 0.47
SLC5A2 P31639 6/20 0.47
HTR6 P50406 1/20 0.46
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PTGS2 P35354 1/20 0.39
KLK7 P49862 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5822476 0.90 KLK7 (0.46) SLC5A1SLC5A2HTR6ALDH1A1MAPT
SCHEMBL5441783 0.84 HTR6 (0.41) SLC5A1SLC5A2HTR6ALDH1A1MAPT
SCHEMBL5432493 0.82 SLC5A1 (0.42) SLC5A1SLC5A2HTR6ALDH1A1MAPT
SCHEMBL5801261 0.81 HTR6 (0.42) SLC5A1SLC5A2HTR6ALDH1A1MAPT
SCHEMBL5240385 0.77 SLC5A1 (0.52) SLC5A1SLC5A2HTR6ALDH1A1MAPT
SCHEMBL5438268 0.76 CRHR1 (0.35) SLC5A1SLC5A2HTR6ALDH1A1MAPT
SCHEMBL4862016 0.72 SLC5A1 (0.49) SLC5A1SLC5A2HTR6ALDH1A1MAPT
Hydrochloric Acid SCHEMBL6134453 0.70 MAPT (0.53) SLC5A1SLC5A2HTR6ALDH1A1MAPT
Hydrochloric Acid SCHEMBL6133263 0.69 HTR6 (0.49) SLC5A1SLC5A2HTR6ALDH1A1MAPT
SCHEMBL5434125 0.66 SLC5A1 (0.40) SLC5A1SLC5A2HTR6MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2006-05-10 EP disclosed
WO-2005019208-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2005-03-03 WO disclosed