SCHEMBL5804157

SCHEMBL5804157

CON(C(N)=O)c1ccc(N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 6/20 0.41
CYP3A4 P08684 6/20 0.41
ALDH1A1 P00352 5/20 0.41
MAPK1 P28482 3/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 4/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
PSMD14 O00487 1/20 0.38
RECQL P46063 1/20 0.38
GFER P55789 1/20 0.38
PARP10 Q53GL7 1/20 0.37
CYP1A2 P05177 3/20 0.36
MAOA P21397 2/20 0.36
LMNA P02545 2/20 0.36
F2 P00734 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
PHLPP2 Q6ZVD8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6037528 0.84 ALOX5 (0.42) TDP1ALDH1A1TP53ALOX15TSHR
SCHEMBL13871569 0.82 RAB9A (0.42) TDP1CYP3A4ALDH1A1TSHRL3MBTL1
SCHEMBL6037494 0.82 NPSR1 (0.41) TDP1CYP3A4ALDH1A1TSHRL3MBTL1
SCHEMBL2895073 0.78 CA1 (0.31) PARP10CA1CA2
SCHEMBL13734403 0.72 ALDH1A1 (0.52) TDP1CYP3A4ALDH1A1MAPK1TP53
SCHEMBL65464 0.72 ALDH1A1 (0.44) TDP1CYP3A4ALDH1A1MAPK1TP53
SCHEMBL11297057 0.71 CYP3A4 (0.41) TDP1CYP3A4ALDH1A1MAPK1TP53
SCHEMBL23246120 0.71 HCAR2 (0.34) ALDH1A1KDM4E
SCHEMBL9233431 0.70 ALDH1A1 (0.42) TDP1CYP3A4ALDH1A1MAPK1TP53
SCHEMBL16706030 0.69 TDP1 (0.52) TDP1CYP3A4ALDH1A1MAPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615925-A1 IMIDAZOPYRIDINE DERIVATIVES AS MELANOCORTIN RECEPTOR AGONISTS Société de Conseils de Recherches et d'Applications Scientifiques ( S.C.R.A.S.) (FR) 2006-01-18 EP disclosed
EP-1599167-A2 NOVEL BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES AND USE THEREOF AS A MEDICAMENT Société de Conseils de Recherches et d'Applications Scientifiques ( S.C.R.A.S.) (FR) 2005-11-30 EP disclosed
WO-2004089951-A1 IMIDAZOPYRIDINE DERIVATIVES HAVING AN AFFINITY FOR MELANOCORTIN RECEPTORS SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2004-10-21 WO disclosed
WO-2004075823-A2 NOVEL BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES AND USE THEREOF AS A MEDICAMENT SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2004-09-10 WO disclosed