SCHEMBL5804272

SCHEMBL5804272

Cc1nc(-c2ccccc2)c(NC(=O)NS(=O)(=O)c2cc3ccccc3s2)s1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 9/20 0.62
FBP1 P09467 1/20 0.45
KIT P10721 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
MALT1 Q9UDY8 1/20 0.41
CA2 P00918 1/20 0.39
HDAC1 Q13547 1/20 0.39
MCL1 Q07820 1/20 0.37
ACP1 P24666 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5815111 0.82 MALT1 (0.41) NTRK1FBP1KITALDH1A1KDM4E
SCHEMBL5813841 0.79 NTRK1 (0.60) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL16595137 0.79 NTRK1 (1.00) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL5804817 0.78 NTRK1 (0.59) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL5815917 0.78 NTRK1 (0.65) NTRK1ALDH1A1KDM4EGAAMAPT
SCHEMBL14148480 0.78 KDR (0.44) FBP1KITALDH1A1KDM4EMAPT
SCHEMBL5813435 0.78 NTRK1 (0.58) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL5801916 0.78 NTRK1 (0.58) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL5814366 0.77 NTRK1 (0.57) NTRK1FBP1ALDH1A1KDM4EPOLB
SCHEMBL5804820 0.76 NTRK1 (0.58) NTRK1ALDH1A1KDM4EPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006085815-A1 THIAZOLE DERIVATIVES, THEIR PROCESS FOR THEIR PREPARATION AND THEIR USE IN THERAPY ASTRAZENECA AB (SE) 2006-08-17 WO disclosed
WO-2006085815-A1 THIAZOLE DERIVATIVES, THEIR PROCESS FOR THEIR PREPARATION AND THEIR USE IN THERAPY ASTRAZENECA AB (SE) 2006-08-17 WO disclosed