SCHEMBL5804435

SCHEMBL5804435

CC(C)[Si](O)(O)C=Cc1ccc(CC(=O)N(CCc2ccccc2)CCc2c[nH]c3ccccc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC5R P33032 7/20 0.49
MC3R P41968 7/20 0.49
HDAC1 Q13547 6/20 0.49
HDAC3 O15379 4/20 0.49
HDAC4 P56524 4/20 0.49
HDAC7 Q8WUI4 4/20 0.49
HDAC2 Q92769 4/20 0.49
HDAC10 Q969S8 4/20 0.49
HDAC11 Q96DB2 4/20 0.49
HDAC8 Q9BY41 4/20 0.49
HDAC6 Q9UBN7 4/20 0.49
HDAC9 Q9UKV0 4/20 0.49
HDAC5 Q9UQL6 4/20 0.49
KCNH2 Q12809 4/20 0.49
MC4R P32245 4/20 0.49
KMT2A Q03164 2/20 0.46
TAAR1 Q96RJ0 1/20 0.46
MEN1 O00255 1/20 0.46
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5804658 0.85 HDAC1 (0.59) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL5807471 0.85 HDAC1 (0.52) MC3RHDAC1HDAC3HDAC4HDAC7
SCHEMBL5805627 0.83 CDK4 (0.48) MC5RMC3RHDAC1HDAC3HDAC4
SCHEMBL5804438 0.82 HDAC1 (0.49) MC5RMC3RHDAC1HDAC3HDAC4
SCHEMBL5807879 0.79 KMT2A (0.55) MC5RMC3RMC4RKMT2ATAAR1
SCHEMBL5807825 0.79 TRPM8 (0.53) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL5804661 0.77 HDAC1 (0.54) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL5806021 0.75 CDK4 (0.44) MC5RMC3RHDAC1HDAC3HDAC4
SCHEMBL5808553 0.73 CDK4 (0.53) HTR1AADRA2AADRA2BADRA2CMAOA
SCHEMBL5804585 0.73 HDAC1 (0.59) HDAC1HDAC3HDAC4HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006069096-A1 SILANOL DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE PHARMACYCLICS, INC. (US) 2006-06-29 WO disclosed