SCHEMBL5805000

SCHEMBL5805000

NC(=O)N(CCCl)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2A1 Q16548 1/20 0.43
CYP3A4 P08684 4/20 0.43
ALDH1A1 P00352 3/20 0.36
ALOX15 P16050 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HIF1A Q16665 2/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36
OPRM1 P35372 2/20 0.36
ABCB11 O95342 1/20 0.36
CHRM2 P08172 1/20 0.36
ADRA2A P08913 1/20 0.36
CHRM1 P11229 1/20 0.36
ACHE P22303 1/20 0.36
PTGS1 P23219 1/20 0.36
DRD3 P35462 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27575737 0.84 CYP3A4 (0.43) BCL2A1CYP3A4ALDH1A1MEN1MAPT
Hydrochloric Acid SCHEMBL10535649 0.82 CYP3A4 (0.50) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
Hydrochloric Acid SCHEMBL27840267 0.81 POLB (0.46) CYP3A4OPRM1TDP1
Hydrochloric Acid SCHEMBL28795770 0.76 ALDH1A1 (0.44) CYP3A4ALDH1A1SMN1; SMN2MAPTKDM4E
SCHEMBL7593179 0.74 EGFR (0.36) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL6517580 0.74 BCL2A1 (0.41) BCL2A1CYP3A4ALDH1A1ALOX15SMN1; SMN2
SCHEMBL2792176 0.74 BCL2A1 (0.46) BCL2A1CYP3A4ALDH1A1SMN1; SMN2HIF1A
SCHEMBL8216746 0.72 L3MBTL1 (0.39) BCL2A1CYP3A4ALDH1A1MEN1KMT2A
SCHEMBL11504229 0.72 BCL2A1 (0.46) BCL2A1CYP3A4ALDH1A1MEN1MAPT
SCHEMBL27419401 0.71 DGAT1 (0.45) ALDH1A1SMN1; SMN2MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed