SCHEMBL5807016

SCHEMBL5807016

O=C(O)NCCCCCCNc1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.50
SLC6A3 Q01959 2/20 0.45
KCNH3 Q9ULD8 2/20 0.44
PRSS1 P07477 4/20 0.43
F2 P00734 2/20 0.43
PRSS2 P07478 2/20 0.43
PRSS3 P35030 2/20 0.43
TMPRSS6 Q8IU80 2/20 0.43
ST14 Q9Y5Y6 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HDAC3 O15379 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
MAPT P10636 1/20 0.42
FOLH1 Q04609 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5305735 1.00 KMT2A (0.50) KMT2ASLC6A3KCNH3PRSS1F2
SCHEMBL5791704 0.98 KMT2A (0.51) KMT2ASLC6A3KCNH3PRSS1NPC1
SCHEMBL19133490 0.95 KMT2A (0.48) KMT2ASLC6A3PRSS1NPC1RAB9A
SCHEMBL25205776 0.84 PRSS1 (0.46) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL25257367 0.84 PRSS1 (0.46) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL29582367 0.81 NPC1 (0.65) NPC1RAB9AHDAC3HDAC1HDAC2
SCHEMBL19133511 0.80 MGLL (0.48) KMT2APRSS1F2PRSS2PRSS3
SCHEMBL19133486 0.80 ALDH1A1 (0.47) KMT2APRSS1MAPTALDH1A1GLA
SCHEMBL19133521 0.80 MAPT (0.57) KMT2ASLC6A3RAB9AMAPTALDH1A1
SCHEMBL28239490 0.80 LMNA (0.53) KMT2AHDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed