Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | HIF1A | Q16665 | 1/20 | 0.34 |
| ▸ | EPAS1 | Q99814 | 1/20 | 0.34 |
| ▸ | CES2 | O00748 | 2/20 | 0.32 |
| ▸ | CES1 | P23141 | 2/20 | 0.32 |
| ▸ | LMNA | P02545 | 1/20 | 0.32 |
| ▸ | MAPT | P10636 | 2/20 | 0.32 |
| ▸ | NPC1 | O15118 | 2/20 | 0.32 |
| ▸ | RAB9A | P51151 | 2/20 | 0.32 |
| ▸ | POLB | P06746 | 1/20 | 0.32 |
| ▸ | MEN1 | O00255 | 1/20 | 0.32 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.32 |
| ▸ | KDM4E | B2RXH2 | 1/20 | 0.31 |
| ▸ | ALDH1A1 | P00352 | 2/20 | 0.31 |
| ▸ | CYP3A4 | P08684 | 1/20 | 0.31 |
| ▸ | ROCK2 | O75116 | 1/20 | 0.30 |
| ▸ | TSHR | P16473 | 1/20 | 0.30 |
| ▸ | MAPK1 | P28482 | 1/20 | 0.30 |
| ▸ | HTT | P42858 | 1/20 | 0.30 |
| ▸ | ATM | Q13315 | 1/20 | 0.30 |
| ▸ | NPY5R | Q15761 | 1/20 | 0.30 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL1682170 | 0.88 | HIF1A (0.33) | HIF1AEPAS1CES2CES1LMNA | |
| SCHEMBL7638594 | 0.85 | HIF1A (0.37) | HIF1AEPAS1CES2CES1LMNA | |
| SCHEMBL9751520 | 0.83 | POLB (0.30) | MAPTNPC1RAB9APOLBMEN1 | |
| SCHEMBL9094342 | 0.83 | MDM2 (0.35) | LMNAMEN1KMT2AALDH1A1CYP3A4 | |
| SCHEMBL8583697 | 0.78 | HIF1A (0.32) | HIF1AEPAS1CES2CES1LMNA | |
| SCHEMBL8818025 | 0.76 | TSHR (0.37) | HIF1AEPAS1CES2CES1LMNA | |
| SCHEMBL4629214 | 0.74 | HIF1A (0.32) | HIF1AEPAS1 | |
| SCHEMBL3984769 | 0.73 | ALDH1A1 (0.36) | HIF1AEPAS1CES2CES1LMNA | |
| SCHEMBL8982590 | 0.73 | ALDH1A1 (0.36) | HIF1AEPAS1CES2CES1LMNA | |
| SCHEMBL27513098 | 0.73 | ALDH1A1 (0.36) | HIF1AEPAS1CES2CES1LMNA |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-3094639-A1 | METHOD FOR OPTIMIZING POST-TRANSLATIONAL MODIFICATIONS ON RECOMBINANT PROTEINS | Leszcyniecka, Magdalena (US) | 2016-11-23 | — | — | EP | disclosed |
| WO-2015106276-A1 | METHOD FOR OPTIMIZING POST-TRANSLATIONAL MODIFICATIONS ON RECOMBINANT PROTEINS | LESZCYNIECKA MAGDALENA (US) | 2015-07-16 | — | — | WO | disclosed |
| WO-2006127842-A2 | TRACERS FOR MONITORING THE ACTIVITY OF SODIUM/GLUCOSE COTRANSPORTERS IN HEALTH AND DISEASE | THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) | 2006-11-30 | — | — | WO | disclosed |
| US-6468688-B2 | CHARGING, DISCHARGING EFFICIENCY; VANADIUM ELECTROLYTE | PINNACLE VRB LIMITED (AU) | 2002-10-22 | — | — | US | disclosed |
| US-20010028977-A1 | Charging, discharging efficiency; vanadium electrolyte | JD HOLDING INC. (KY) | 2001-10-11 | — | — | US | disclosed |
| EP-0428605-A1 | SYNTHETIC RECEPTOR ANALOGUES. | SYMBICOM AB (SE) | 1991-05-29 | — | — | EP | disclosed |
| WO-1990001488-A1 | SYNTHETIC RECEPTOR ANALOGUES | SYMBICOM AKTIEBOLAG (SE) | 1990-02-22 | — | — | WO | disclosed |