SCHEMBL5808086

SCHEMBL5808086

CCCOC(=O)[C@H](C)c1c(C)n(C(=O)c2ccc(Cl)c(F)c2)c2cc(F)c(O)c(F)c12

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.36
SMYD3 Q9H7B4 1/20 0.33
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
IDO1 P14902 1/20 0.31
KCNH2 Q12809 1/20 0.31
TSHR P16473 1/20 0.30
TACR2 P21452 1/20 0.30
TACR1 P25103 1/20 0.30
TACR3 P29371 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5808087 1.00 PTGS2 (0.36) PTGS2SMYD3AKR1C3AKR1C2IDO1
SCHEMBL5813384 0.95 PTGS2 (0.38) PTGS2TSHR
SCHEMBL5813388 0.95 PTGS2 (0.38) PTGS2TSHR
SCHEMBL5797882 0.94 PTGS2 (0.36) PTGS2SMYD3TSHR
SCHEMBL5797881 0.94 PTGS2 (0.36) PTGS2SMYD3TSHR
SCHEMBL5800660 0.93 PTGS2 (0.37) PTGS2AKR1C3AKR1C2
SCHEMBL5800661 0.93 PTGS2 (0.37) PTGS2AKR1C3AKR1C2
SCHEMBL5798596 0.91 PTGS2 (0.44) PTGS2AKR1C3AKR1C2
SCHEMBL5798592 0.91 PTGS2 (0.44) PTGS2AKR1C3AKR1C2
SCHEMBL5809647 0.90 PTGS2 (0.37) PTGS2SMYD3AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed