SCHEMBL5808194

SCHEMBL5808194

Cc1ccc(-n2nc(C(=O)NC3CCCc4ccccc43)c3c2CCCC3)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.54
USP2 O75604 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C19 P33261 1/20 0.54
HTT P42858 1/20 0.54
UGCG Q16739 1/20 0.52
TAS1R3 Q7RTX0 5/20 0.52
TAS1R1 Q7RTX1 5/20 0.52
TAS1R2 Q8TE23 4/20 0.52
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 1/20 0.49
POLB P06746 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
TSHR P16473 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5811315 0.91 CNR1 (0.55) LMNAUSP2CYP1A2CYP3A4CYP2D6
SCHEMBL14003135 0.77 HTT (0.52) LMNAHTTTAS1R3TAS1R1TAS1R2
SCHEMBL5807932 0.74 UGCG (0.53) UGCGMEN1KMT2ACNR1CNR2
SCHEMBL5822464 0.74 CNR2 (0.85) UGCGCNR1CNR2
SCHEMBL5808694 0.71 CNR2 (0.68) UGCGMEN1KMT2ACNR1CNR2
SCHEMBL5812049 0.69 CNR1 (0.69) LMNAUGCGALDH1A1CNR1CNR2
SCHEMBL19554499 0.69 ALDH1A1 (0.54) LMNAHTTTAS1R3TAS1R1TAS1R2
SCHEMBL13545818 0.69 DHODH (0.66) HTTTAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL342298 0.69 GAA (0.49) LMNAUSP2CYP1A2CYP3A4CYP2D6
SCHEMBL342297 0.69 GAA (0.49) LMNAUSP2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006030124-A1 CONDENSED PYRAZOLE DERIVATIVES, PREPARATION METHOD THEREOF AND THERAPEUTIC USE OF SAME SANOFI-AVENTIS (FR) 2006-03-23 WO claimed