SCHEMBL5808246

SCHEMBL5808246

Cc1cc2nc(NCC(=Cc3ccc(C(=O)NO)cc3)CCOc3cccc4ccccc34)sc2cc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 2/20 0.42
HDAC1 Q13547 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
MCL1 Q07820 5/20 0.37
PIN1 Q13526 3/20 0.37
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37
CSNK2A3 Q8NEV1 1/20 0.37
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5808243 1.00 P2RX3 (0.42) P2RX3HDAC1HDAC6HDAC3HDAC4
SCHEMBL5823606 0.92 PIN1 (0.40) P2RX3MCL1PIN1CSNK2A2CSNK2B
SCHEMBL5809988 0.89 SCD (0.46) HDAC1MCL1MAPTMEN1KMT2A
SCHEMBL5809983 0.89 SCD (0.46) HDAC1MCL1MAPTMEN1KMT2A
SCHEMBL5799747 0.86 MAPT (0.44) P2RX3MCL1MAPTMEN1KMT2A
SCHEMBL5799742 0.86 MAPT (0.44) P2RX3MCL1MAPTMEN1KMT2A
SCHEMBL5798801 0.83 HDAC1 (0.38) P2RX3HDAC1HDAC6HDAC3HDAC4
SCHEMBL5810050 0.82 P2RX3 (0.49) P2RX3HDAC1HDAC6HDAC3HDAC4
SCHEMBL5810052 0.82 P2RX3 (0.49) P2RX3HDAC1HDAC6HDAC3HDAC4
SCHEMBL5797931 0.81 P2RX3 (0.45) P2RX3HDAC1HDAC6HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006025683-A1 ARYLAMINOMETHYL PROPENYL BENZHYDROXYAMID DERIVATIVES WITH INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-03-09 WO disclosed