SCHEMBL5808272

SCHEMBL5808272

O=Cc1cnn(-c2ccccc2)c1-c1cc(F)cc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
NPSR1 Q6W5P4 2/20 0.44
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
POLB P06746 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HIF1A Q16665 2/20 0.40
HTT P42858 1/20 0.40
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
NR3C1 P04150 1/20 0.38
S1PR1 P21453 1/20 0.38
MGLL Q99685 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
USP2 O75604 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL673658 0.79 HIF1A (0.42) LMNANPSR1NPC1RAB9APOLB
SCHEMBL5730469 0.74 PTGS2 (0.45) LMNANPSR1HIF1APTGS2PTGS1
SCHEMBL2649068 0.70 RAB9A (0.54) NPC1RAB9APOLBALDH1A1MEN1
SCHEMBL1566534 0.70 MAPK1 (0.54) LMNANPC1RAB9AALDH1A1PTGS2
SCHEMBL3321144 0.70 RAB9A (0.49) LMNANPSR1NPC1RAB9AALDH1A1
SCHEMBL13407215 0.70 NR4A3 (0.44) LMNANPSR1NPC1RAB9APOLB
SCHEMBL28600941 0.70 HIF1A (0.41) LMNANPSR1NPC1RAB9APOLB
SCHEMBL4039361 0.70 MAPT (0.59) LMNANPSR1NPC1RAB9APOLB
SCHEMBL13019208 0.69 PTGS1 (0.43) LMNANPSR1POLBALDH1A1PTGS1
SCHEMBL15330142 0.68 ERN1 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006033995-A2 THIAZOLIDIN-4-ONES HAVING ANTI-HEPATITIS B ACTIVITY VALEANT RESEARCH AND DEVELOPMENT (US) 2006-03-30 WO disclosed