SCHEMBL5809153

SCHEMBL5809153

O=C(NN=CCc1cccc(O)c1)c1cc(Cl)c(O)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCGR P47871 3/20 0.48
SPHK2 Q9NRA0 10/20 0.46
SPHK1 Q9NYA1 8/20 0.43
ADCYAP1R1 P41586 1/20 0.42
CYP2D6 P10635 1/20 0.41
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5815660 1.00 GCGR (0.48) GCGRSPHK2SPHK1ADCYAP1R1CYP2D6
SCHEMBL1669458 0.75 MEN1 (0.53) SPHK2SPHK1ADCYAP1R1NPC1MAPT
SCHEMBL6002241 0.72 POLB (0.47) MAPT
SCHEMBL25620321 0.71 ENPP2 (0.52) MAPT
SCHEMBL11302626 0.70 ALDH1A1 (0.55) NPC1MAPTRAB9A
SCHEMBL17541218 0.70 ALDH1A1 (0.55) NPC1MAPTRAB9A
SCHEMBL5809141 0.70 GAA (0.65) CYP2D6NPC1MAPTRAB9A
SCHEMBL2474636 0.69 SPHK2 (0.47) SPHK2SPHK1NPC1MAPTRAB9A
SCHEMBL22295829 0.68 CYP1A2 (0.42) MAPT
SCHEMBL21211500 0.68 GCGR (0.57) GCGRSPHK2SPHK1CYP2D6NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006136008-A1 SALICYLIC ACID HYDRAZONES AS INHIBITORS OF THE ERK MAPKINASE PATHWAY AND FOR THE TREATMENT OF CANCER UNIVERSITY HEALTH NETWORK (CA) 2006-12-28 WO disclosed