SCHEMBL5811323

SCHEMBL5811323

O=C(Nc1ccccc1)c1cccc(F)c1C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.60
KMT2A Q03164 5/20 0.60
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
TDP1 Q9NUW8 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.56
LMNA P02545 3/20 0.55
ALDH1A1 P00352 1/20 0.53
HTT P42858 2/20 0.53
P2RX1 P51575 2/20 0.52
KCNK3 O14649 1/20 0.52
KCNK9 Q9NPC2 1/20 0.52
P2RX7 Q99572 1/20 0.52
HPGD P15428 2/20 0.51
KDM4E B2RXH2 1/20 0.51
TP53 P04637 1/20 0.51
HSD17B10 Q99714 1/20 0.51
TLR8 Q9NR97 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
PTGS1 P23219 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27928793 0.87 MEN1 (0.55) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL28799328 0.83 PTGS1 (0.62) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL4363732 0.81 MEN1 (0.89) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL30739691 0.80 KMT2A (0.68) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL9343198 0.79 KMT2A (0.66) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL31388520 0.78 ALB (0.57) ALDH1A1P2RX1P2RX7HPGDKDM4E
SCHEMBL1259459 0.78 ALB (0.57) ALDH1A1P2RX1P2RX7HPGDKDM4E
SCHEMBL28995015 0.78 KMT2A (0.64) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL8535595 0.77 KCNK3 (0.62) KMT2AKCNK3KCNK9HPGDRXFP1
SCHEMBL22820183 0.77 NPC1 (0.67) MEN1KMT2ANPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006086229-A1 THE USE OF SELECTIVE P2X7 RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2006-08-17 WO disclosed