SCHEMBL22820183

SCHEMBL22820183

O=C(Nc1ccccc1)c1cccc(C(=O)Nc2ccc(C(F)(F)F)cc2)c1F

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.67
RAB9A P51151 2/20 0.67
PTGS1 P23219 2/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
RXFP1 Q9HBX9 5/20 0.56
LMNA P02545 1/20 0.56
P2RX1 P51575 1/20 0.56
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
MTOR P42345 1/20 0.55
KCNK3 O14649 2/20 0.55
KCNK9 Q9NPC2 1/20 0.55
TDP1 Q9NUW8 1/20 0.54
GPR27 Q9NS67 1/20 0.54
EPHX2 P34913 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12700361 0.84 NPC1 (0.71) NPC1RAB9APTGS1SMN1; SMN2RXFP1
SCHEMBL22819939 0.84 LMNA (0.70) NPC1RAB9ALMNAMEN1KMT2A
SCHEMBL22819966 0.82 ALDH1A1 (0.70) NPC1RAB9ASMN1; SMN2LMNAMEN1
SCHEMBL22820200 0.81 NPC1 (0.64) NPC1RAB9ASMN1; SMN2LMNAMEN1
SCHEMBL2698258 0.81 P2RX1 (0.75) NPC1RAB9APTGS1SMN1; SMN2LMNA
SCHEMBL2638776 0.81 PTGS1 (0.70) NPC1RAB9APTGS1SMN1; SMN2RXFP1
SCHEMBL30665186 0.81 P2RX1 (0.75) NPC1RAB9APTGS1SMN1; SMN2LMNA
SCHEMBL31393757 0.81 CHRNB2 (0.71) NPC1RAB9APTGS1SMN1; SMN2
SCHEMBL2564890 0.80 NPC1 (1.00) NPC1RAB9APTGS1LMNAP2RX1
SCHEMBL4247052 0.80 NPC1 (0.86) NPC1RAB9APTGS1LMNAP2RX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020255425-A1 ANTI-HBV AGENT 国立研究開発法人理化学研究所 2020-12-24 WO disclosed