SCHEMBL5811883

SCHEMBL5811883

CCC(CO)NC.Cc1cc(F)ccc1[C@H]1CCCN1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.43
JAK2 O60674 1/20 0.41
NTRK1 P04629 1/20 0.41
HSP90AA1 P07900 2/20 0.39
HSP90AB1 P08238 2/20 0.39
GRM5 P41594 2/20 0.38
RIPK1 Q13546 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6064294 0.81 TACR1 (0.54) TACR1HSP90AA1HSP90AB1GRM5RIPK1
SCHEMBL6064290 0.81 TACR1 (0.54) TACR1HSP90AA1HSP90AB1GRM5RIPK1
SCHEMBL6550098 0.80 TACR1 (0.53) TACR1HSP90AA1HSP90AB1GRM5RIPK1
SCHEMBL30145299 0.76 TACR1 (0.52) TACR1HSP90AA1HSP90AB1GRM5RIPK1
SCHEMBL6311676 0.75 TACR1 (0.36) TACR1JAK2NTRK1
SCHEMBL6311681 0.75 TACR1 (0.36) TACR1JAK2NTRK1
SCHEMBL5811888 0.75 TACR1 (0.36) TACR1JAK2NTRK1
Maleic Acid SCHEMBL30145281 0.73 TACR1 (0.47) TACR1GRM5RIPK1
SCHEMBL5414345 0.72 TACR1 (0.44) TACR1
SCHEMBL4021108 0.72 TACR1 (0.64) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638935-A1 NK1 ANTAGONIST Pfizer Products Inc. (US) 2006-03-29 EP disclosed
WO-2004110996-A1 NK1 ANTAGONIST PFIZER PRODUCTS INC. (US) 2004-12-23 WO disclosed