SCHEMBL5812487

SCHEMBL5812487

C[C@](N)(c1ccccc1)c1nccc(-c2scnc2-c2cccc(Cl)c2)n1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.39
ADORA1 P30542 7/20 0.39
RORB Q92753 2/20 0.38
TGFBR1 P36897 1/20 0.38
KMO O15229 1/20 0.37
ADORA2B P29275 3/20 0.37
PLK1 P53350 1/20 0.36
DPP4 P27487 1/20 0.36
CYP19A1 P11511 1/20 0.35
IDO1 P14902 1/20 0.34
PIM1 P11309 1/20 0.34
CDK4 P11802 1/20 0.34
CDK2 P24941 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819107 0.88 ADORA2A (0.38) ADORA2AADORA1KMOADORA2BDPP4
SCHEMBL5813644 0.82 CCNT1 (0.47) ADORA2AADORA1TGFBR1KMOPLK1
SCHEMBL5817990 0.82 PTGDR2 (0.36) ADORA2AADORA1TGFBR1MAPK14
SCHEMBL5821649 0.80 ADORA2A (0.39) ADORA2AADORA1DPP4CYP19A1MAPK14
SCHEMBL5819868 0.78 CDC7 (0.38) ADORA2AADORA1TGFBR1DPP4PIM1
SCHEMBL5820844 0.77 KCNH2 (0.41) TGFBR1MAPK14
SCHEMBL5820628 0.77 KCNH2 (0.46)
SCHEMBL5818662 0.76 KCNH2 (0.44) MAPK14
SCHEMBL5818860 0.76 LMNA (0.44) ADORA2AADORA1RORBTGFBR1KMO
SCHEMBL5812491 0.76 CAMK2D (0.47) PLK1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO claimed