SCHEMBL7522368

SCHEMBL7522368

COc1ccc(CNc2nc(-c3ccncc3)nc3scc(C)c23)cc1OC.Cc1csc2nc(-c3ccncc3)nc(Cl)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ESR1 P03372 1/20 0.46
TNF P01375 1/20 0.41
NOD1 Q9Y239 1/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
PRKCI P41743 5/20 0.41
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
STAT1 P42224 1/20 0.39
TGFBR1 P36897 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
APP P05067 1/20 0.38
PGK1 P00558 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5119865 0.94 MEN1 (0.52) ALDH1A1MEN1KMT2AESR1TNF
SCHEMBL5814645 0.94 ESR1 (0.46) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL5809020 0.91 ALDH1A1 (0.61) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL5115035 0.90 ESR1 (0.48) MEN1KMT2AESR1PRKCITGFBR1
SCHEMBL5814517 0.86 ESR1 (0.43) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL5813871 0.85 MEN1 (0.46) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL7516802 0.85 ALDH1A1 (0.56) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL5118580 0.84 ALDH1A1 (0.55) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL5120732 0.83 ESR1 (0.53) ESR1ROCK2ROCK1PRKCITGFBR1
SCHEMBL8179394 0.83 MEN1 (0.48) ALDH1A1SMN1; SMN2MEN1KMT2AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920431-A1 THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 1999-06-09 EP disclosed
WO-1998006722-A1 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 1998-02-19 WO disclosed