Fumaric Acid

Fumaric Acid

SCHEMBL5816

O=C([O-])/C=C\C(=O)O.[K+]

nearest known ligand 0.00

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Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL106350 1.00
Maleic Acid SCHEMBL6365123 1.00 TSHR (0.60)
Fumaric Acid SCHEMBL5819 1.00
Fumaric Acid SCHEMBL28720329 0.97 TSHR (0.56)
Fumaric Acid SCHEMBL28032519 0.97 TSHR (0.56)
Fumaric Acid SCHEMBL5250318 0.97 TSHR (0.56)
Fumaric Acid SCHEMBL28384623 0.94 TSHR (0.53)
Fumaric Acid SCHEMBL106909 0.93
Fumaric Acid SCHEMBL106910 0.93
Fumaric Acid SCHEMBL5799074 0.93 TSHR (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2508 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4646583-A1 POTASSIUM MALEATE BUFFER FOR FREE CHLORINE ANALYSIS Hach Company (US) 2025-11-12 EP claimed
US-20240315956-A1 METHOD OF PRODUCTION OF THE COMPOSITION OF CYCLOOXYGENASE-2 (COX-2) INHIBITORS US Nano Food & Drug INC 2024-09-26 US claimed
US-20240230609-A1 POTASSIUM MALEATE BUFFER FOR FREE CHLORINE ANALYSIS HACH COMPANY (US) 2024-07-11 US claimed
WO-2024147903-A1 POTASSIUM MALEATE BUFFER FOR FREE CHLORINE ANALYSIS HACH COMPANY (US) 2024-07-11 WO claimed
EP-3481878-B1 AMINE COMPOSITION USEFUL FOR MAKING POLYURETHANE FOAM EVONIK OPERATIONS GMBH (DE) 2024-05-22 EP claimed
EP-4366732-A1 METHOD OF PRODUCTION OF THE COMPOSITION OF CYCLOOXYGENASE-2 (COX-2) INHIBITORS US Nano Food & Drug Inc (US) 2024-05-15 EP claimed
CN-117813089-A Process for producing cyclooxygenase-2 (COX-2) inhibitor composition 美国纳米食品药品公司 2024-04-02 CN claimed
WO-2023281449-A1 METHOD OF PRODUCTION OF THE COMPOSITION OF CYCLOOXYGENASE-2 (COX-2) INHIBITORS US Nano Food & Drug INC (US) 2023-01-12 WO claimed
CN-109476803-B Amine compositions useful for making polyurethane foams 赢创运营有限公司 2022-04-12 CN claimed
US-11021561-B2 Amine composition useful for making polyurethane foam EVONIK OPERATIONS GMBH (DE) 2021-06-01 US claimed
EP-0831706-B1 NON-AQUEOUS COMPOSITIONS CONTAINING A HALOALKYNYL COMPOUND AND A BUFFER FOR PROVIDING BIOCIDAL ACTIVITY AND FOR STABILIZING END-USE FORMULATIONS TROY TECHNOLOGY CORP INC (US) 2003-05-02 EP claimed
US-6124350-A PAINT CONTAINING A BIOCIDAL COMPOSITION COMPRISING A HALOPROPYNYL COMPOUND AND A BUFFER TROY TECHNOLOGY CORPORATION, INC. (US) 2000-09-26 US claimed
US-6017955-A A BUFFER STABILIZER FOR ADJUSTING THE PH OF END-USE FORMULATION BETWEEN 3.0 AND 8.0 TO PREVENT DEGRADATION OF PESTICIDE 3-IODO-2-PROPYNYL BUTYL CARBAMATE TROY TECHNOLOGY CORPORATION, INC. (US) 2000-01-25 US claimed
EP-0831706-A1 METHOD OF STABILIZING BIOCIDAL COMPOSITIONS OF HALOALKYNYL COMPOUNDS TROY CHEMICAL CORPORATION (US) 1998-04-01 EP claimed
EP-0578451-B1 Process for preparing polysuccinimide polymers ROHM & HAAS (US) 1998-01-14 EP claimed
WO-1996039836-A1 METHOD OF STABILIZING BIOCIDAL COMPOSITIONS OF HALOALKYNYL COMPOUNDS TROY CHEMICAL COMPANY (US) 1996-12-19 WO claimed
US-5371179-A Polysuccinimide polymers and process for preparing polysuccinimide polymers ROHM AND HAAS COMPANY (US) 1994-12-06 US claimed
EP-0578451-A2 Polysuccinimide polymers and process for preparing polysuccinimide polymers ROHM AND HAAS COMPANY (US) 1994-01-12 EP claimed
US-4668735-A MONOSODIUM, MONOPOTASSIUM, MONOAMMONIUM MALEATE; SOLUTION POLYMERIZATION KAO CORPORATION (JP) 1987-05-26 US claimed
US-4061465-A Creasable durable press textiles from methylol reagents and half amides or half salts of dicarboxylic acids THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF AGRICULTURE (US) 1977-12-06 US claimed