SCHEMBL5817145

SCHEMBL5817145

COc1ccc2c(c1)c(CC(=O)NCCCO[N+](=O)[O-])c(C)n2CC1CCCCC1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 5/20 0.63
PTGS2 P35354 13/20 0.62
PTGS1 P23219 8/20 0.62
HRH4 Q9H3N8 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA4 P22748 1/20 0.45
CA9 Q16790 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5815957 0.81 PTGS2 (0.64) PLA2G2APTGS2PTGS1CA12CA1
SCHEMBL7952544 0.79 PLA2G2A (0.82) PLA2G2APTGS2PTGS1
SCHEMBL7952825 0.78 PLA2G2A (1.00) PLA2G2APTGS2
SCHEMBL5806528 0.76 PTGS2 (1.00) PTGS2PTGS1HRH4CA12CA1
SCHEMBL7968767 0.76 PLA2G2A (0.78) PLA2G2APTGS2
SCHEMBL5808472 0.74 PLA2G2A (0.73) PLA2G2APTGS2PTGS1
SCHEMBL5808467 0.69 PTGS2 (0.42) PTGS2PTGS1
SCHEMBL12106622 0.68 PTGS2 (0.84) PTGS2PTGS1HRH4CA12CA1
SCHEMBL5820566 0.68 PTGS2 (1.00) PTGS2PTGS1HRH4CA12CA1
SCHEMBL5106790 0.67 PTGS2 (0.75) PTGS2PTGS1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006099416-A1 2-METHYL INDOLE CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2006-09-21 WO claimed
WO-2006099416-A1 2-METHYL INDOLE CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2006-09-21 WO disclosed