SCHEMBL5819216

SCHEMBL5819216

COc1cc2c(cc1OC)-c1c(c3cc(C(F)(F)F)ccc3n1CC(=O)NCCCCCCN)CC(=O)N2

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 10/20 0.47
CCNB2 O95067 9/20 0.47
CCNB1 P14635 9/20 0.47
GSK3B P49841 9/20 0.47
CCNB3 Q8WWL7 9/20 0.47
CDK5 Q00535 6/20 0.47
CDK5R1 Q15078 6/20 0.47
SMYD3 Q9H7B4 1/20 0.37
PLK1 P53350 1/20 0.36
KMT2A Q03164 1/20 0.34
MAPT P10636 2/20 0.33
GAA P10253 1/20 0.33
CRBN Q96SW2 1/20 0.33
MPO P05164 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5813979 0.99 CDK1 (0.47) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5806193 0.89 CDK1 (0.56) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5802551 0.87 CDK1 (0.51) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5802944 0.85 CDK1 (0.46) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5815923 0.84 CDK1 (0.56) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5823198 0.82 CDK1 (0.57) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5814486 0.79 CDK1 (0.57) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5802955 0.79 CDK1 (0.53) CDK1CCNB2CCNB1GSK3BCCNB3
Hydrochloric Acid SCHEMBL5803457 0.79 CDK1 (0.57) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5819011 0.75 CDK1 (0.55) CDK1CCNB2CCNB1GSK3BCCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006089874-A1 BENZO[2,3]AZEPINO[4,5-B]INDOL-6-ONES GPC BIOTECH AG (DE) 2006-08-31 WO claimed