SCHEMBL5819963

SCHEMBL5819963

Cc1cc(Cl)c(OCCOc2ccc(C3=C(C(=O)O)C4CC[C@@H](C3)N4C(=O)OC(C)(C)C)cc2)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.43
REN P00797 10/20 0.40
CYP3A4 P08684 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.36
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819961 1.00 ATM (0.43) ATMRENCYP3A4L3MBTL1SLC6A4
SCHEMBL5668307 0.89 REN (0.41) ATMRENCYP3A4
SCHEMBL5668304 0.89 REN (0.41) ATMRENCYP3A4
SCHEMBL1752405 0.89 REN (0.41) ATMRENCYP3A4
SCHEMBL2473476 0.81 REN (0.44) RENCYP3A4KCNH2
SCHEMBL12750478 0.80 REN (0.39) ATMRENCYP3A4L3MBTL1
SCHEMBL4785962 0.80 REN (0.63) RENCYP3A4
SCHEMBL4785977 0.80 REN (0.63) RENCYP3A4
SCHEMBL4785966 0.80 REN (0.63) RENCYP3A4
SCHEMBL1751812 0.79 NPBWR1 (0.39) L3MBTL1SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1680427-A1 DIAZABICYCLONONENE AND TETRAHYDROPYRIDINE DERIVATIVES AS RENIN INHIBITORS Actelion Pharmaceuticals Ltd. (CH) 2006-07-19 EP disclosed
WO-2005040173-A1 DIAZABICYCLONONENE AND TETRAHYDROPYRIDINE DERIVATIVES AS RENIN INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2005-05-06 WO disclosed