SCHEMBL5820076

SCHEMBL5820076

COC(=O)CCc1nccc(C)c1NC(C)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
HSD17B10 Q99714 3/20 0.40
HPGD P15428 2/20 0.40
PTPRB P23467 1/20 0.40
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
HTT P42858 2/20 0.36
JAK2 O60674 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
TSHR P16473 1/20 0.35
EGFR P00533 2/20 0.35
LMNA P02545 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16919139 0.73 ALDH1A1 (0.49) KDM4EHSD17B10HPGDPTPRBALDH1A1
SCHEMBL1345232 0.73 GAA (0.42) KDM4EHSD17B10HPGDPTPRBALDH1A1
SCHEMBL24455228 0.72 NOS2 (0.40) KDM4EHSD17B10ALDH1A1SMN1; SMN2HTT
SCHEMBL28781635 0.71 HPGD (0.37) HSD17B10HPGDPTPRBALDH1A1SMN1; SMN2
SCHEMBL19475136 0.71 GAA (0.45) KDM4EHSD17B10HPGDPTPRBALDH1A1
SCHEMBL6952630 0.70 NR3C2 (0.52)
SCHEMBL27955096 0.70 ATR (0.53) KDM4EEGFR
SCHEMBL23373281 0.70 NR3C2 (0.42) KDM4EHSD17B10ALDH1A1TSHRLMNA
SCHEMBL8825478 0.69 ALDH1A1 (0.53) KDM4EHSD17B10HPGDALDH1A1SMN1; SMN2
SCHEMBL31048845 0.69 LMNA (0.45) KDM4EALDH1A1SMN1; SMN2TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670798-A1 AMINOPYRIDINE-DERIVATIVES AS INDUCTIBLE NO-SYNTHASE INHIBITORS Altana Pharma AG (DE) 2006-06-21 EP disclosed
WO-2005061496-A1 AMINOPYRIDINE-DERIVATIVES AS INDUCTIBLE NO-SYNTHASE INHIBITORS ALTANA PHARMA AG (DE) 2005-07-07 WO disclosed