SCHEMBL5820439

SCHEMBL5820439

CSc1nc(Nc2ccc(N3CCOCC3)cc2)cc(N2CCN(CC(=O)N3CCN(c4ccccc4O)CC3)CC2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.44
CYP1A2 P05177 1/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
RECQL P46063 1/20 0.42
NPC1 O15118 2/20 0.42
GAA P10253 1/20 0.41
ALOX15 P16050 1/20 0.41
RAB9A P51151 2/20 0.41
AURKA O14965 2/20 0.40
AURKB Q96GD4 1/20 0.40
MAPT P10636 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
IGF1R P08069 1/20 0.40
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ZAP70 P43403 1/20 0.38
HPGD P15428 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820251 0.91 CYP1A2 (0.45) NAMPTCYP1A2ALDH1A1KDM4ERECQL
SCHEMBL5821064 0.90 SMN1; SMN2 (0.44) NAMPTCYP1A2ALDH1A1KDM4ENPC1
SCHEMBL5820813 0.90 NAMPT (0.47) NAMPTCYP1A2ALDH1A1KDM4ERECQL
SCHEMBL5823980 0.89 ZAP70 (0.49) NAMPTCYP1A2ALDH1A1KDM4ERECQL
SCHEMBL5823039 0.89 AURKA (0.50) NAMPTCYP1A2ALDH1A1KDM4ERECQL
SCHEMBL5816069 0.87 AURKA (0.43) NAMPTCYP1A2ALDH1A1KDM4ERECQL
SCHEMBL5821753 0.86 AURKA (0.45) NAMPTCYP1A2NPC1RAB9AAURKA
SCHEMBL5815028 0.86 RAB9A (0.46) NAMPTCYP1A2NPC1RAB9AAURKA
SCHEMBL5821823 0.85 JAK3 (0.42) NAMPTCYP1A2ALDH1A1KDM4ERECQL
SCHEMBL5823587 0.85 JAK2 (0.43) NAMPTCYP1A2NPC1RAB9AAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137706-A1 6-(4-SUBSTITUTED-ANILINO)PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM. CO., LTD. (KR) 2006-12-28 WO claimed
WO-2006137706-A1 6-(4-SUBSTITUTED-ANILINO)PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM. CO., LTD. (KR) 2006-12-28 WO disclosed