SCHEMBL5821138

SCHEMBL5821138

O=C(O)CC[C@H]([AsH2])Cc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPA3 P15088 2/20 0.62
KEAP1 Q14145 1/20 0.55
NAALAD2 Q9Y3Q0 2/20 0.53
FFAR1 O14842 2/20 0.52
SLC15A1 P46059 1/20 0.51
LTA4H P09960 1/20 0.49
CYP1A2 P05177 2/20 0.48
CPA1 P15085 2/20 0.47
CPB1 P15086 1/20 0.47
CPB2 Q96IY4 1/20 0.47
HDAC3 O15379 1/20 0.47
MAPK1 P28482 1/20 0.47
ADRA1A P35348 1/20 0.47
HDAC4 P56524 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HDAC1 Q13547 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20512303 0.80 CPA3 (0.60) CPA3KEAP1FFAR1SLC15A1LTA4H
SCHEMBL10710074 0.80 CPA3 (0.67) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL6495926 0.78 CPA3 (0.65) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL6502909 0.78 CPA3 (0.65) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL6495924 0.78 CPA3 (0.65) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL5767750 0.77 CPA3 (0.62) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL288473 0.77 CPA3 (0.62) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL757260 0.77 CPA3 (0.62) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL3440803 0.77 CPA3 (0.62) CPA3KEAP1NAALAD2FFAR1SLC15A1
SCHEMBL3963424 0.77 CPA3 (1.00) CPA3NAALAD2CYP1A2CPA1CPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620432-A1 NK-2 ANTAGONIST BASIC LINEAR COMPOUNDS AND FORMULATIONS CONTAINING THEM Menarini Ricerche S.p.A. (IT) 2006-02-01 EP disclosed
WO-2004094412-A1 NK-2 ANTAGONIST BASIC LINEAR COMPOUNDS AND FORMULATIONS CONTAINING THEM MENARINI RICERCHE S.P.A. (IT) 2004-11-04 WO disclosed