SCHEMBL5821175

SCHEMBL5821175

CNC(=N)c1c(SC)n(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccccc2)nc1=O

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
PTGS2 P35354 12/20 0.41
PTGS1 P23219 2/20 0.39
CHRNA7 P36544 1/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
GRM5 P41594 1/20 0.38
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819681 0.92 CA9 (0.43) KMT2AGAACA12CA1CA2
SCHEMBL5822322 0.92 CA9 (0.43) KMT2AGAACA12CA1CA2
SCHEMBL5815528 0.91 GAA (0.38) KMT2AGAACA12CA1CA2
SCHEMBL5817765 0.90 CA1 (0.44) CA12CA1CA2CA9PTGS2
SCHEMBL5821439 0.90 CA9 (0.44) KMT2AGAACA12CA1CA2
SCHEMBL5815486 0.89 PTGS2 (0.39) KMT2AGAACA12CA1CA2
SCHEMBL5821281 0.88 PTGS2 (0.38) KMT2AGAACA12CA1CA2
SCHEMBL5821767 0.81 ESR1 (0.36) GAAPTGS2PTGS1
SCHEMBL5820891 0.79 ALDH1A1 (0.41) GAAPTGS2PTGS1
SCHEMBL5821417 0.77 ALDH1A1 (0.36) KMT2AMEN1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO claimed
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed