SCHEMBL5815528

SCHEMBL5815528

CNC(=N)c1c(SC)n(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccncc2)nc1=O

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
CA2 P00918 10/20 0.38
CA1 P00915 9/20 0.38
CA9 Q16790 9/20 0.38
CA12 O43570 8/20 0.38
PTGS2 P35354 6/20 0.37
CYP2D6 P10635 1/20 0.33
PTGS1 P23219 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5822322 0.91 CA9 (0.43) GAAKMT2ACA2CA1CA9
SCHEMBL5821175 0.91 KMT2A (0.47) GAAKMT2ACA2CA1CA9
SCHEMBL5819681 0.91 CA9 (0.43) GAAKMT2ACA2CA1CA9
SCHEMBL5817765 0.90 CA1 (0.44) CA2CA1CA9CA12PTGS2
SCHEMBL5821439 0.89 CA9 (0.44) GAAKMT2ACA2CA1CA9
SCHEMBL5815486 0.88 PTGS2 (0.39) GAAKMT2ACA2CA1CA9
SCHEMBL5821281 0.87 PTGS2 (0.38) GAAKMT2ACA2CA1CA9
SCHEMBL5815685 0.86 AOC3 (0.41) GAAKMT2A
SCHEMBL5821417 0.86 ALDH1A1 (0.36) KMT2A
SCHEMBL5820968 0.85 CA2 (0.38) GAAKMT2ACA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed