SCHEMBL5821792

SCHEMBL5821792

CC(C)(C)OC(=O)N(C(=O)NCc1ccccc1)c1ccco1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA7 P43166 1/20 0.41
CA14 Q9ULX7 1/20 0.41
ATM Q13315 1/20 0.40
PPARA Q07869 1/20 0.40
RAB9A P51151 3/20 0.40
POLB P06746 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 2/20 0.40
RIPK1 Q13546 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10853381 0.78 CTDSP1 (0.44) SMN1; SMN2MEN1KMT2AHPGDTSHR
SCHEMBL5033374 0.76 CTDSP1 (0.50) SMN1; SMN2MEN1KMT2AHPGDTSHR
SCHEMBL4193440 0.76 CA12 (0.47) SMN1; SMN2HPGDTSHRCA12CA1
SCHEMBL4246502 0.75 CA12 (0.46) SMN1; SMN2HPGDCA12CA1CA7
SCHEMBL29140328 0.72 NPC1 (0.42) SMN1; SMN2MEN1KMT2ARAB9APOLB
SCHEMBL13430486 0.71 OPRM1 (0.44) SMN1; SMN2HPGDCA12CA1CA7
SCHEMBL216618 0.70 NPC1 (0.41) SMN1; SMN2MEN1KMT2ATSHRRAB9A
SCHEMBL10795492 0.70 SMN1; SMN2 (0.37) SMN1; SMN2MEN1KMT2AHPGDTSHR
SCHEMBL3838871 0.70 CA12 (0.63) SMN1; SMN2MEN1KMT2ACA12CA1
SCHEMBL4246507 0.69 AKT1 (0.53) CA12CA1CA7CA14ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465896-A4 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2006-01-11 EP disclosed
EP-1465896-A2 MITOTIC KINESIN INHIBITORS Merck & Co., Inc. (US) 2004-10-13 EP disclosed
WO-2003050122-A2 MITOTIC KINESIN INHIBITORS MERCK & CO., INC. (US) 2003-06-19 WO disclosed