SCHEMBL582599

SCHEMBL582599

CCOC(=O)CC(=O)C1CCN(C(=O)OC)C(c2ccc(C(F)(F)F)nc2)C1.COC(=O)N1CCC(C(=O)O)CC1c1ccc(C(F)(F)F)nc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.35
PSEN1 P49768 6/20 0.34
PSEN2 P49810 6/20 0.34
APH1B Q8WW43 6/20 0.34
NCSTN Q92542 6/20 0.34
APH1A Q96BI3 6/20 0.34
PSENEN Q9NZ42 6/20 0.34
TRPM8 Q7Z2W7 1/20 0.33
FPR1 P21462 1/20 0.33
FPR2 P25090 1/20 0.33
EGLN2 Q96KS0 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
EGLN3 Q9H6Z9 1/20 0.33
EPHX2 P34913 1/20 0.33
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
KCNQ4 P56696 1/20 0.33
KCNQ5 Q9NR82 1/20 0.33
HDAC4 P56524 1/20 0.33
SSTR1 P30872 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL582600 1.00 HRH3 (0.35) HRH3PSEN1PSEN2APH1BNCSTN
SCHEMBL3075597 0.97 HRH3 (0.37) HRH3PSEN1PSEN2APH1BNCSTN
SCHEMBL581198 0.97 HRH3 (0.37) HRH3PSEN1PSEN2APH1BNCSTN
SCHEMBL3085403 0.97 HRH3 (0.37) HRH3PSEN1PSEN2APH1BNCSTN
SCHEMBL581335 0.89 HRH3 (0.41) HRH3PSEN1PSEN2APH1BNCSTN
SCHEMBL581726 0.87 NOTUM (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL581727 0.87 NOTUM (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL582439 0.83 ALDH1A1 (0.36)
SCHEMBL582438 0.83 ALDH1A1 (0.36)
SCHEMBL582069 0.83 EPHX2 (0.42) TRPM8EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed