SCHEMBL5828673

SCHEMBL5828673

Cc1cc2[nH]c3ccccc3c2c2c1C(=O)NC2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 1.00
CDK4 P11802 8/20 0.61
CCND1 P24385 8/20 0.61
CAMK2B Q13554 6/20 0.61
CAMK2G Q13555 6/20 0.61
CAMK2D Q13557 6/20 0.61
CAMK2A Q9UQM7 6/20 0.61
CCNE2 O96020 6/20 0.61
CCNE1 P24864 6/20 0.61
CDK2 P24941 6/20 0.61
CDK5 Q00535 3/20 0.61
CDK5R1 Q15078 3/20 0.61
CCNB2 O95067 3/20 0.61
CDK1 P06493 3/20 0.61
CCNB1 P14635 3/20 0.61
CCNB3 Q8WWL7 3/20 0.61
CCNA2 P20248 2/20 0.61
MEN1 O00255 1/20 0.61
PRKD3 O94806 1/20 0.61
PRKCG P05129 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832547 0.79 WEE1 (0.74) PARP1CDK4CCND1CAMK2BCAMK2G
SCHEMBL9832776 0.77 WEE1 (0.75) PARP1CDK4CCND1CAMK2BCAMK2G
Staurosporine Aglycon SCHEMBL29406635 0.76 CDK4 (1.00) PARP1CDK4CCND1CAMK2BCAMK2G
Staurosporine Aglycon SCHEMBL30530825 0.76 CDK4 (1.00) PARP1CDK4CCND1CAMK2BCAMK2G
Staurosporine Aglycon SCHEMBL8124103 0.76 CDK4 (1.00) PARP1CDK4CCND1CAMK2BCAMK2G
SCHEMBL10405623 0.76 WEE1 (0.76) PARP1CAMK2DCDK2CDK5CDK1
SCHEMBL9832075 0.76 WEE1 (0.77) PARP1CDK4CCND1CAMK2BCAMK2G
SCHEMBL22566985 0.75 CDK4 (0.74) PARP1CDK4CCND1CAMK2BCAMK2G
SCHEMBL29516962 0.74 PARP1 (1.00) PARP1CDK4CCND1CAMK2BCAMK2G
SCHEMBL5381581 0.74 PARP1 (1.00) PARP1CDK4CCND1CAMK2BCAMK2G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US disclosed