SCHEMBL582882

SCHEMBL582882

CCOC(=O)CC(=O)[C@H]1CCN(C)[C@H](Cc2cc(F)ccc2F)C1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
CHRM3 P20309 13/20 0.40
DPP4 P27487 3/20 0.39
DPP7 Q9UHL4 3/20 0.39
DPP8 Q6V1X1 2/20 0.39
DPP9 Q86TI2 2/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3080101 0.87 ALDH1A1 (0.42) ALDH1A1TDP1DPP4DPP7DPP8
SCHEMBL3076465 0.87 ALDH1A1 (0.42) ALDH1A1TDP1DPP4DPP7DPP8
SCHEMBL581683 0.87 ALDH1A1 (0.42) ALDH1A1TDP1DPP4DPP7DPP8
SCHEMBL3075396 0.80 ALDH1A1 (0.49) ALDH1A1TDP1KDM4EMEN1KMT2A
SCHEMBL581488 0.80 ALDH1A1 (0.49) ALDH1A1TDP1KDM4EMEN1KMT2A
SCHEMBL3081361 0.80 ALDH1A1 (0.49) ALDH1A1TDP1KDM4EMEN1KMT2A
SCHEMBL582364 0.80 HTR2A (0.41) ALDH1A1MEN1KMT2A
SCHEMBL582160 0.77 KMT2A (0.41) ALDH1A1TDP1KDM4EMEN1KMT2A
SCHEMBL581942 0.76 KMT2A (0.37) ALDH1A1CHRM3KDM4EMEN1KMT2A
SCHEMBL581773 0.75 ALDH1A1 (0.43) ALDH1A1TDP1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed