SCHEMBL582364

SCHEMBL582364

CCOC(=O)CC(=O)[C@H]1CCN(C)[C@H](CCc2ccc(F)cc2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.41
HTR2C P28335 2/20 0.41
HTR7 P34969 2/20 0.41
HTR6 P50406 2/20 0.41
GRM2 Q14416 3/20 0.40
CACNA1G O43497 2/20 0.40
ALDH1A1 P00352 3/20 0.39
RECQL P46063 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
OPRM1 P35372 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
CHRM1 P11229 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
CCR3 P51677 1/20 0.38
SLC6A3 Q01959 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581334 0.87 CACNA1G (0.38) HTR2AHTR2CHTR7HTR6GRM2
SCHEMBL3085356 0.87 CACNA1G (0.38) HTR2AHTR2CHTR7HTR6GRM2
SCHEMBL581333 0.87 CACNA1G (0.38) HTR2AHTR2CHTR7HTR6GRM2
SCHEMBL586938 0.84 FFAR4 (0.37) HTR2AHTR2CHTR7HTR6GRM2
SCHEMBL586937 0.84 FFAR4 (0.37) HTR2AHTR2CHTR7HTR6GRM2
SCHEMBL582160 0.81 KMT2A (0.41) ALDH1A1OPRM1CHRM1MEN1KMT2A
SCHEMBL582882 0.80 ALDH1A1 (0.44) ALDH1A1MEN1KMT2A
SCHEMBL3075222 0.78 PPARG (0.40) ALDH1A1RECQLOPRM1CHRM1MEN1
SCHEMBL582086 0.78 PPARG (0.40) ALDH1A1RECQLOPRM1CHRM1MEN1
SCHEMBL3075705 0.78 PPARG (0.40) ALDH1A1RECQLOPRM1CHRM1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed