SCHEMBL5835754

SCHEMBL5835754

CSC(C)c1cnc(N)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.43
BACE1 P56817 1/20 0.37
MYC P01106 1/20 0.36
WDR5 P61964 1/20 0.36
ALDH1A1 P00352 3/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
GRM8 O00222 1/20 0.33
GRM4 Q14833 1/20 0.33
MAPT P10636 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CSNK2A1 P68400 1/20 0.32
PTGER3 P43115 1/20 0.31
POLB P06746 2/20 0.31
THRB P10828 1/20 0.31
HTT P42858 1/20 0.31
RECQL P46063 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL682219 0.79
SCHEMBL5875737 0.75
SCHEMBL23153450 0.73 SLC6A3 (0.33)
SCHEMBL5875764 0.71 NOS1 (0.42) NOS1BACE1MYCWDR5ALDH1A1
SCHEMBL5119808 0.69 NOS1 (0.45) NOS1BACE1MYCWDR5ALDH1A1
SCHEMBL5029681 0.69 GRM8 (0.47) NOS1BACE1ALDH1A1HPGDALOX15
SCHEMBL12877806 0.69 NOS1 (0.41) NOS1BACE1ALDH1A1HPGDALOX15
SCHEMBL25921275 0.68 APLNR (0.30)
SCHEMBL17643502 0.68 KMT2A (0.53) NOS1BACE1ALDH1A1HPGDGRM8
SCHEMBL12877375 0.68 NOS1 (0.39) NOS1BACE1MYCWDR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037929-B1 2-amino-thiazole derivatives, process for their preparation, and their use as antitumor agents PHARMACIA & UPJOHN S.P.A. (IT) 2006-05-02 US disclosed