SCHEMBL5837100

SCHEMBL5837100

CC(=O)NC(C(=O)NCC1OCCc2c1sc(NC(=O)C(=O)OC(C)(C)C)c2C(=O)OC(C)(C)C)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 7/20 0.36
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPRB P23467 1/20 0.34
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
POLB P06746 1/20 0.32
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6315778 0.88 PTPN2 (0.38) CXCR2PTPN2PTPN1PTPRBALDH1A1
SCHEMBL5841311 0.86 CTSS (0.32) CXCR2ALDH1A1HPGDPOLBCTSS
SCHEMBL5838379 0.86 CTSS (0.32) CXCR2ALDH1A1HPGDPOLBCTSS
SCHEMBL5838437 0.83 CTSS (0.38) CXCR2PTPN2PTPN1PTPRBCTSS
SCHEMBL5842479 0.82 PTPN1 (0.45) PTPN2PTPN1PTPRBPOLB
SCHEMBL5837519 0.82 PTPN1 (0.45) PTPN2PTPN1PTPRBPOLB
SCHEMBL5837475 0.81 PTPN1 (0.40) CXCR2PTPN2PTPN1PTPRBALDH1A1
SCHEMBL5838593 0.80 PTPN2 (0.39) CXCR2PTPN2PTPN1PTPRBALDH1A1
SCHEMBL5838097 0.80 CTSS (0.45) CXCR2CTSSCTSK
SCHEMBL5837704 0.76 CXCR2 (0.39) CXCR2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115624-B1 Method of inhibiting protein tyrosine phosphatase 1B and/or T-cell protein tyrosine phosphatase 4 and/or other PTPases with an Asp residue at position 48 NOVO NORDISK A/S (DK) 2006-10-03 US disclosed