SCHEMBL5838653

SCHEMBL5838653

Cc1nc(-c2ccccn2)ccc1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
ALDH1A1 P00352 4/20 0.47
NNMT P40261 1/20 0.47
KDM4E B2RXH2 7/20 0.47
LMNA P02545 3/20 0.47
CCR1 P32246 2/20 0.47
CCR5 P51681 2/20 0.47
CCR8 P51685 2/20 0.47
TP53 P04637 2/20 0.47
ALOX15 P16050 2/20 0.47
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
ALPL P05186 1/20 0.47
HSP90AA1 P07900 1/20 0.47
ALPI P09923 1/20 0.47
ALPG P10696 1/20 0.47
MAPK1 P28482 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10169399 0.81 NPSR1 (0.45) NPSR1RXFP1ALDH1A1KDM4ELMNA
SCHEMBL22584043 0.79 GRM5 (0.51) NPSR1RXFP1ALDH1A1KDM4EALOX15
SCHEMBL2815367 0.77 NPSR1 (0.47) NPSR1RXFP1ALDH1A1KDM4EGRM5
SCHEMBL18765298 0.76 NPSR1 (0.46) NPSR1RXFP1ALDH1A1KDM4ELMNA
SCHEMBL29933397 0.76 PARP1 (0.67) NPSR1RXFP1KDM4ELMNACCR1
SCHEMBL11927613 0.74 KDM4E (0.59) NPSR1ALDH1A1KDM4ELMNACCR1
SCHEMBL22468488 0.74 BTK (0.46) NPSR1RXFP1KDM4ELMNACCR1
SCHEMBL22468497 0.74 BTK (0.58) NPSR1RXFP1ALDH1A1KDM4ETP53
SCHEMBL12272145 0.74 NNMT (0.46) RXFP1ALDH1A1NNMTSMN1; SMN2BTK
SCHEMBL935065 0.73 KDM4E (0.59) NPSR1RXFP1ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732566-A2 6-AZAINDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2006-12-20 EP disclosed
WO-2005097129-A2 6-AZAINDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-10-20 WO disclosed