SCHEMBL5840892

SCHEMBL5840892

O=S1(=O)N[C]Nc2cc(Cl)sc21

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCC8 Q09428 12/20 0.47
KCNJ11 Q14654 12/20 0.47
GRIA1 P42261 3/20 0.36
GRIA2 P42262 3/20 0.36
GRIA3 P42263 3/20 0.36
GRIA4 P48058 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3870329 0.68 GRIA1 (0.46) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL8473189 0.68 ABCC8 (0.57) ABCC8KCNJ11
SCHEMBL4256373 0.62 ABCC8 (0.49) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL6792625 0.61 ABCC8 (0.44) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL6208560 0.61 ABCC8 (0.38) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL10542378 0.59 RET (0.44) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL6798761 0.59 ABCC8 (0.43) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL8286612 0.59 ABCC8 (0.50) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL6997132 0.59 ABCC8 (0.43) ABCC8KCNJ11GRIA1GRIA2GRIA3
SCHEMBL13536240 0.57 GRIA1 (0.45) ABCC8KCNJ11GRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214325-B1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK AS (DK) 2005-11-09 EP claimed
EP-1214325-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2002-06-19 EP claimed
WO-2001019831-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2001-03-22 WO claimed
US-7019026-B1 Modulators of Protein Tyrosine Phosphatases (PTPases) NOVO NORDISK A/S (DK) 2006-03-28 US disclosed
EP-1214325-B1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK AS (DK) 2005-11-09 EP disclosed
EP-1214325-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2002-06-19 EP disclosed
WO-2001019831-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2001-03-22 WO disclosed