SCHEMBL5843192

SCHEMBL5843192

CC(NC(=O)C(O)c1ccccc1)C(N)=O

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.52
NFE2L2 Q16236 1/20 0.52
LMNA P02545 4/20 0.47
MAPK1 P28482 1/20 0.47
PSMB5 P28074 1/20 0.46
NAAA Q02083 2/20 0.45
MME P08473 2/20 0.44
HPGD P15428 1/20 0.43
CTRB1 P17538 2/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ALOX5 P09917 1/20 0.42
KDM1A O60341 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27896435 1.00 KEAP1 (0.52) KEAP1NFE2L2LMNAMAPK1PSMB5
SCHEMBL5843204 1.00 KEAP1 (0.52) KEAP1NFE2L2LMNAMAPK1PSMB5
SCHEMBL15743807 0.84 KEAP1 (0.54) KEAP1NFE2L2LMNAMAPK1PSMB5
SCHEMBL8584122 0.84 CTSD (0.56) LMNAMMEMEN1KMT2A
SCHEMBL8584123 0.84 CTSD (0.56) LMNAMMEMEN1KMT2A
SCHEMBL197183 0.82 KEAP1 (0.58) KEAP1NFE2L2LMNAMAPK1PSMB5
SCHEMBL197182 0.82 KEAP1 (0.58) KEAP1NFE2L2LMNAMAPK1PSMB5
SCHEMBL28408400 0.80 MEN1 (0.64) KEAP1NFE2L2LMNAMAPK1HPGD
SCHEMBL8974575 0.80 MEN1 (0.64) KEAP1NFE2L2LMNAMAPK1HPGD
SCHEMBL19119737 0.80 KEAP1 (0.50) KEAP1NFE2L2LMNAMAPK1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102791693-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2012-11-21 CN claimed
US-7109243-B2 Inhibitors of cathepsin S IRM LLC (BM) 2006-09-19 US claimed