SCHEMBL5847231

SCHEMBL5847231

CC(C)(C)OC(=O)N1CC[C@@H]2[C@H](C1)c1cc(Br)cc3c1N2CCCC3=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.41
USP30 Q70CQ3 3/20 0.39
FPR2 P25090 3/20 0.37
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.36
PDE4B Q07343 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
EPHX1 P07099 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847677 0.87 NPC1 (0.41) GPR119USP30FPR2IDO1TDO2
SCHEMBL5846934 0.87 NPC1 (0.41) GPR119USP30FPR2IDO1TDO2
SCHEMBL5410957 0.85 HTR2A (0.36) MAPTKDM4EHTR2AHTR2CMEN1
SCHEMBL5410954 0.85 HTR2A (0.36) MAPTKDM4EHTR2AHTR2CMEN1
SCHEMBL5848121 0.84 NPC1 (0.40) GPR119USP30FPR2IDO1TDO2
SCHEMBL5847390 0.84 FPR2 (0.42) GPR119USP30FPR2IDO1TDO2
SCHEMBL5847999 0.84 NPC1 (0.40) GPR119USP30FPR2IDO1TDO2
SCHEMBL5848322 0.84 NPC1 (0.40) GPR119USP30FPR2IDO1TDO2
SCHEMBL5848240 0.84 GPR119 (0.42) GPR119USP30HPGDHTR2AHTR2C
SCHEMBL5848252 0.83 USP30 (0.41) GPR119USP30FPR2IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed