SCHEMBL5848601

SCHEMBL5848601

Cc1cc(C#N)ccc1-c1cc2c3c(c1)[C@@H]1CN(C(=O)OC(C)(C)C)CC[C@@H]1N3CCC2

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
GPR119 Q8TDV5 9/20 0.40
ALK Q9UM73 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PTK2 Q05397 1/20 0.36
CETP P11597 4/20 0.36
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
RET P07949 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848913 1.00 HTR2A (0.41) HTR2AHTR2CHTR2BGPR119ALK
SCHEMBL5847204 0.98 GPR119 (0.40) HTR2AHTR2CHTR2BGPR119ALK
SCHEMBL5407323 0.88 HTR2A (0.41) HTR2AHTR2CHTR2BHRH2HRH1
SCHEMBL6918350 0.88 HTR2A (0.41) HTR2AHTR2CHTR2BHRH2HRH1
SCHEMBL5847313 0.87 HTR2A (0.51) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5410813 0.86 HTR2A (0.39) HTR2AHTR2CHTR2BHRH2HRH1
SCHEMBL5848103 0.85 HTR2A (0.49) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5847114 0.82 HTR2A (0.45) HTR2AHTR2CHTR2BGPR119
SCHEMBL5848567 0.82 HTR2C (0.41) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5849712 0.81 USP30 (0.39) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed