SCHEMBL5849709

SCHEMBL5849709

COc1ccc(-c2cccc(C)c2)cc1N

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.63
CYP3A4 P08684 2/20 0.63
HTR2C P28335 1/20 0.51
TSHR P16473 2/20 0.50
HSD17B10 Q99714 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
RAB9A P51151 2/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
APP P05067 1/20 0.49
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
KMT2A Q03164 1/20 0.47
GAA P10253 1/20 0.46
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6492701 0.86 ALDH1A1 (0.71) ALDH1A1CYP3A4HTR2CTSHRHSD17B10
SCHEMBL30839809 0.84 ALDH1A1 (0.67) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL31607677 0.84 ALDH1A1 (0.67) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL6863931 0.84 ALDH1A1 (0.67) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL3783522 0.84 ALDH1A1 (0.52) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL330530 0.83 ALDH1A1 (0.55) ALDH1A1CYP3A4HTR2CTSHRHSD17B10
Hydrochloric Acid SCHEMBL1143402 0.81 ALDH1A1 (0.55) ALDH1A1CYP3A4HTR2CTSHRHSD17B10
SCHEMBL5835015 0.81 ALOX5 (0.62) ALDH1A1TSHRHSD17B10TDP1RAB9A
SCHEMBL8264634 0.79 CD274 (0.49) ALDH1A1HTR2CTSHRHSD17B10RAB9A
SCHEMBL55544 0.78 ALDH1A1 (1.00) ALDH1A1CYP3A4TSHRHSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1306131-B1 Cross-coupling process using a catalyst comprising a cyclic nitrogen ligand SUMITOMO CHEMICAL CO (JP) 2016-12-07 EP disclosed
US-20060111593-A1 Coupling catalyst and process using the same SUMITOMO CHEMICAL COMPANY, LIMITED 2006-05-25 US disclosed
US-7041856-B2 Coupling catalyst and process using the same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-05-09 US disclosed
US-20030162950-A1 Coupling catalyst and process using the same SUMITOMO CHEMICAL COMPANY, LIMITED 2003-08-28 US disclosed
EP-1306131-A2 Cross-Coupling catalyst comprising a cyclic nitrogen ligand and process using the same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-05-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030162950-A1 Coupling catalyst and process using the same NOD1, PYM1, C9 ALDH1A1 3293/4885CYP3A4 2291/4885HTR2C 2262/4885
US-20060111593-A1 Coupling catalyst and process using the same RPL22, C9, RBM22 ALDH1A1 3723/4885CYP3A4 1666/4885HTR2C 921/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.