SCHEMBL585060

SCHEMBL585060

O=Cc1cnc(-c2cccs2)s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.53
KDM4E B2RXH2 8/20 0.42
ALDH1A1 P00352 6/20 0.42
HSD17B10 Q99714 2/20 0.42
EPHX2 P34913 1/20 0.42
RAB9A P51151 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 2/20 0.40
MEN1 O00255 1/20 0.40
CASP3 P42574 1/20 0.40
KMT2A Q03164 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
ERN1 O75460 1/20 0.37
POLB P06746 1/20 0.37
CYP2A6 P11509 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL585682 0.91 DPP4 (0.64) DPP4KDM4EALDH1A1HSD17B10EPHX2
SCHEMBL584121 0.91 DPP4 (0.64) DPP4KDM4EALDH1A1HSD17B10EPHX2
SCHEMBL869424 0.77 KDM4E (0.50) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL17099921 0.77 ALDH1A1 (0.48) KDM4EALDH1A1MAPTTDP1CYP2A6
SCHEMBL3072249 0.76 KDM4E (0.48) DPP4KDM4EALDH1A1HSD17B10EPHX2
SCHEMBL13722983 0.73 KDM4E (0.36) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL27688648 0.73 KDM4E (0.38) DPP4KDM4EALDH1A1HSD17B10EPHX2
SCHEMBL867509 0.73 KDM4E (0.46) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL9394 0.73 ALDH1A1 (0.50) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL10690511 0.73 KDM4E (0.47) KDM4EALDH1A1HSD17B10EPHX2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10431745-B2 Diketopyrrolopyrrole polymers for use in organic field effect transistors BASF SE (DE) 2019-10-01 US disclosed
EP-3456756-A2 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC FIELD EFFECT TRANSISTORS BASF SE (DE) 2019-03-20 EP disclosed
US-10224484-B2 Diketopyrrolopyrrole polymers for use in organic field effect transistors BASF SE (DE) 2019-03-05 US disclosed
US-20190027690-A9 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC FIELD EFFECT TRANSISTORS BASF SE (DE) 2019-01-24 US disclosed
EP-2350160-B1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC SEMICONDUCTOR DEVICES BASF SE (DE) 2018-04-11 EP disclosed
US-9893288-B2 Diketopyrrolopyrrole polymers for use in organic field effect transistors BASF SE (DE) 2018-02-13 US disclosed
US-9893288-B2 Diketopyrrolopyrrole polymers for use in organic field effect transistors BASF SE (DE) 2018-02-13 US disclosed
US-20170148992-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC FIELD EFFECT TRANSISTORS BASF SE (DE) 2017-05-25 US disclosed
US-20170148991-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC FIELD EFFECT TRANSISTORS BASF SE (DE) 2017-05-25 US disclosed
US-20170148991-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC FIELD EFFECT TRANSISTORS BASF SE (DE) 2017-05-25 US disclosed
US-20110240981-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC FIELD EFFECT TRANSISTORS BASF SE (DE) 2011-10-06 US disclosed
US-20110215313-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC SEMICONDUCTOR DEVICES BASF SE (DE) 2011-09-08 US disclosed
US-20110215313-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC SEMICONDUCTOR DEVICES BASF SE (DE) 2011-09-08 US disclosed
WO-2010115767-A1 PYRROLOPYRROLE DERIVATIVES, THEIR MANUFACTURE AND USE AS SEMICONDUCTORS BASF SE (DE) 2010-10-14 WO disclosed
WO-2010115767-A1 PYRROLOPYRROLE DERIVATIVES, THEIR MANUFACTURE AND USE AS SEMICONDUCTORS BASF SE (DE) 2010-10-14 WO disclosed
WO-2010080864-A1 PIPERIDINE-CONTAINING COMPOUNDS AND USE THEREOF ARRAY BIOPHARMA INC. (US) 2010-07-15 WO disclosed
WO-2010080864-A1 PIPERIDINE-CONTAINING COMPOUNDS AND USE THEREOF ARRAY BIOPHARMA INC. (US) 2010-07-15 WO disclosed
WO-2010049323-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC SEMICONDUCTOR DEVICES BASF SE (DE) 2010-05-06 WO disclosed
WO-2010049321-A1 DIKETOPYRROLOPYRROLE POLYMERS FOR USE IN ORGANIC FIELD EFFECT TRANSISTORS BASF SE (DE) 2010-05-06 WO disclosed
CN-1465567-A Dihydropyridone derivative and use thereof 陈依军 2004-01-07 CN disclosed