SCHEMBL5852274

SCHEMBL5852274

Cc1ccc(S(=O)(=O)N(C)C2(C(=O)N[C@@H](Cc3ccc(NC(=O)c4ccccc4Br)cc3)C(=O)O)CCCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 17/20 0.51
ITGA4 P13612 17/20 0.51
MMP9 P14780 1/20 0.46
ITGB7 P26010 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5851025 0.93 CA1 (0.45) ITGB1ITGA4MMP9ITGB7
SCHEMBL5850857 0.86 ITGB1 (0.64) ITGB1ITGA4ITGB7
SCHEMBL7401948 0.85 ITGB1 (0.61) ITGB1ITGA4MMP9ITGB7
SCHEMBL5850609 0.84 MMP9 (0.49) ITGB1ITGA4MMP9ITGB7
SCHEMBL5851039 0.79 ATM (0.55) ITGB1ITGA4ITGB7
SCHEMBL5850976 0.79 ITGB1 (0.47) ITGB1ITGA4MMP9ITGB7
SCHEMBL7409938 0.78 ATM (0.55) ITGB1ITGA4ITGB7
SCHEMBL5850545 0.77 ITGB1 (0.52) ITGB1ITGA4ITGB7
SCHEMBL5850678 0.77 USP30 (0.44) ITGB1ITGA4MMP9
SCHEMBL6714274 0.76 ITGB1 (0.65) ITGB1ITGA4MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP claimed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-7030114-B1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-04-18 US disclosed