SCHEMBL5854887

SCHEMBL5854887

COC(=O)C(CCCCCCCCC1c2ccc(OC)cc2SCC1(C)c1ccc(OC)cc1)(CCCC(F)(F)C(F)(F)F)C(=O)OC

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.32
MTNR1B P49286 7/20 0.32
NQO2 P16083 6/20 0.32
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7128086 1.00 MTNR1A (0.32) MTNR1AMTNR1BNQO2GAA
SCHEMBL5854225 0.93 ALDH1A1 (0.33)
SCHEMBL5854319 0.93 MTNR1A (0.31) MTNR1AMTNR1BNQO2
SCHEMBL7813218 0.91 SIGMAR1 (0.32)
SCHEMBL5856235 0.87
SCHEMBL6940319 0.87 ESR1 (0.33) MTNR1AMTNR1BNQO2
SCHEMBL7087556 0.87 ESR1 (0.33) MTNR1AMTNR1BNQO2
SCHEMBL5856061 0.85 ESR1 (0.40) MTNR1AMTNR1BNQO2
SCHEMBL5854915 0.85 ESR1 (0.40) MTNR1AMTNR1BNQO2
SCHEMBL5855627 0.84 MTNR1A (0.32) MTNR1AMTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074819-B2 Benzopyran or thiobenzopyran derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2006-07-11 US disclosed
US-6645951-B1 Antiestrogens for treating breast cancer CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-11-11 US disclosed
EP-1087959-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-04-04 EP disclosed
WO-1999065893-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES C & C RESEARCH LABORATORIES (KR) 1999-12-23 WO disclosed