SCHEMBL5857960

SCHEMBL5857960

Cc1ccc2c(c1)ncn2C1CCN(CCC(C)c2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.54
SLC6A4 P31645 1/20 0.54
TACR2 P21452 1/20 0.46
CYP2D6 P10635 2/20 0.46
CCR5 P51681 2/20 0.46
FGFR1 P11362 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5858744 0.89 DRD2 (0.68) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5858702 0.88 DRD2 (0.53) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5860221 0.88 SLC6A4 (0.53) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5860217 0.86 DRD2 (0.50) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5858700 0.85 TACR2 (0.52) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5857199 0.85 DRD2 (0.49) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5858680 0.83 DRD2 (0.52) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5860261 0.83 SLC6A4 (0.52) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5857996 0.80 SLC6A4 (0.50) DRD2SLC6A4TACR2CYP2D6CCR5
SCHEMBL5858616 0.78 DRD2 (0.69) DRD2SLC6A4TACR2CYP2D6CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6989393-B2 Ccr5 modulators benzimidazoles or benzotriazoles ASTRAZENECA AB (SE) 2006-01-24 US disclosed