SCHEMBL5860261

SCHEMBL5860261

CC(CCN1CCC(n2cnc3ccc(F)cc32)CC1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.52
DRD2 P14416 1/20 0.52
ALDH1A1 P00352 2/20 0.46
SLC6A2 P23975 2/20 0.45
SLC6A3 Q01959 2/20 0.45
TACR2 P21452 1/20 0.45
CCR5 P51681 2/20 0.42
CYP2D6 P10635 1/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5860221 0.93 SLC6A4 (0.53) SLC6A4DRD2ALDH1A1SLC6A2SLC6A3
SCHEMBL5858680 0.88 DRD2 (0.52) SLC6A4DRD2TACR2CCR5CYP2D6
SCHEMBL5858744 0.87 DRD2 (0.68) SLC6A4DRD2ALDH1A1TACR2CCR5
SCHEMBL5858700 0.85 TACR2 (0.52) SLC6A4DRD2TACR2CCR5CYP2D6
SCHEMBL5857960 0.83 DRD2 (0.54) SLC6A4DRD2TACR2CCR5CYP2D6
SCHEMBL5858702 0.82 DRD2 (0.53) SLC6A4DRD2TACR2CCR5CYP2D6
SCHEMBL5857996 0.82 SLC6A4 (0.50) SLC6A4DRD2SLC6A2SLC6A3TACR2
SCHEMBL5860217 0.80 DRD2 (0.50) SLC6A4DRD2TACR2CCR5CYP2D6
SCHEMBL5857199 0.79 DRD2 (0.49) SLC6A4DRD2TACR2CCR5CYP2D6
SCHEMBL5860215 0.78 TACR2 (0.45) SLC6A4DRD2TACR2CCR5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6989393-B2 Ccr5 modulators benzimidazoles or benzotriazoles ASTRAZENECA AB (SE) 2006-01-24 US disclosed